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A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
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Increased Valency Improves Inhibitory Activity of Peptides Targeting Proprotein Convertase Subtilisin/Kexin Type 9

Benjamin J Tombling1, Carmen Lammi2, Carlotta Bollati2

  • 1Institute for Molecular Bioscience, Australian Research Council Centre of Excellence for Innovations in Peptide and Protein Science, The University of Queensland, Brisbane, Qld, 4072, Australia.

Chembiochem : a European Journal of Chemical Biology
|March 23, 2021
PubMed

Keywords:
PCSK9cell-based activitydrug designinhibitorspeptide-decorated dendrimers

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