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Updated: Nov 4, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Class A G protein-coupled receptors assemble into functional higher-order hetero-oligomers

Xianlong Gao1, Garrett A Enten1,2, Anthony J DeSantis1

  • 1Department of Surgery, Morsani College of Medicine, University of South Florida, Tampa, FL, USA.

FEBS Letters
|May 25, 2021
PubMed

Keywords:
ACKR3AVPR1ACXCR4receptor dimerreceptor hetero-oligomerizationɑ1-adrenergic receptor

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