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Multifunctional Enkephalin Analogs with a New Biological Profile: MOR/DOR Agonism and KOR Antagonism

Yeon Sun Lee1, Michael Remesic2, Cyf Ramos-Colon2

  • 1Department of Pharmacology, University of Arizona, Tucson, AZ 85724, USA.

Biomedicines
|June 2, 2021
PubMed

Keywords:
analgesic effectskappa receptor antagonistsmultifunctional activityopioid receptorspeptidomimeticsplasma stabilitytemplate-based alignment modeling

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