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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers

Eline Sijbesma1, Kenneth K Hallenbeck2, Sebastian A Andrei1

  • 1Laboratory of Chemical Biology, Department of Biomedical Engineering and Institute for Complex Molecular Systems (ICMS), Eindhoven University of Technology, 5600 MB Eindhoven, The Netherlands.

ACS Medicinal Chemistry Letters
|June 17, 2021
PubMed

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