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Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain

Michael Brand1, James Clayton1, Mustafa Moroglu1

  • 1Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.

Journal of Medicinal Chemistry
|July 13, 2021
PubMed
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