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Updated: Oct 18, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Piperazine squaric acid diamides, a novel class of allosteric P2X7 receptor antagonists

Marius Patberg1, Andreas Isaak1, Friederike Füsser2

  • 1European Institute for Molecular Imaging (EIMI), Waldeyerstr. 15, 48149, Münster, Germany.

European Journal of Medicinal Chemistry
|September 27, 2021
PubMed

Keywords:
AllostericAntagonistsP2XP2X7 receptorSquaric acid

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