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Overview of PROTACs Targeting the Estrogen Receptor: Achievements for Biological and Drug Discovery

Hui Qin1, Yiwen Zhang1,2, Yutao Lou3

  • 1Clinical Pharmacy Center, Department of Pharmacy, Zhejiang Provincial People\'s Hospital, Affiliated People\'s Hospital, Hangzhou Medical College, Hangzhou, Zhejiang, 310014, China.

Current Medicinal Chemistry
|November 11, 2021
PubMed

Keywords:
DNA binding regionER-αER-βEstrogen receptors (ERs)PROTACsnuclear receptor (NR)

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