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Amino acids and its pharmaceutical applications: A mini review
Agustina Bongioanni1, Maria Soledad Bueno1, Belén Alejandra Mezzano1
1Unidad de Investigación y Desarrollo en Tecnología Farmacéutica, UNITEFA-CONICET, Departamento de Ciencias Farmacéuticas, Facultad de Ciencias Químicas, Universidad Nacional de Córdoba, Cordoba X5000HUA, Argentina.
Amino acids are safe natural compounds that enhance drug delivery. This review details their formulation methods and proven ability to improve drug solubility, permeation, stabilization, and therapeutic efficacy.
Area of Science:
- Pharmaceutical Sciences
- Drug Delivery
- Biochemistry
Background:
- Amino acids are naturally occurring compounds with established safety profiles.
- There is significant interest in utilizing amino acids within the pharmaceutical industry.
- Understanding amino acid properties is crucial for pharmaceutical applications.
Purpose of the Study:
- To provide a comprehensive overview of recent investigations on amino acids in pharmaceutical applications.
- To describe the preparation and formulation of amino acids for drug delivery.
- To explore the impact of amino acid formulations on drug properties and therapeutic efficacy.
Main Methods:
- Review of recent scientific literature on amino acid applications in pharmaceuticals.
- Description of common methods for preparing amino acid formulations.
- Analysis of studies on amino acid effects on active pharmaceutical ingredients (APIs).
Main Results:
- Amino acids exhibit beneficial properties for pharmaceutical formulations.
- Formulation methods involving amino acids can enhance API solubilization, permeation, and stabilization.
- Multicomponent systems utilizing amino acids show promise.
Conclusions:
- Amino acids can significantly improve the biopharmaceutical properties of drugs.
- The use of amino acids in drug formulations offers a viable strategy to enhance therapeutic efficacy.
- Further research into amino acid-based drug delivery systems is warranted.
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