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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Pharmacological Effect of GABA Analogues on GABA-ϱ2 Receptors and Their Subtype Selectivity

Moawiah M Naffaa1, David E Hibbs1, Mary Chebib1

  • 1School of Pharmacy, Faculty of Medicine and Health, University of Sydney, Sydney, NSW 2006, Australia.

Life (Basel, Switzerland)
|January 21, 2022
PubMed

Keywords:
GABA analoguesGABA-ϱ subtype-selectivityGABA-ϱ2 receptorsadditive/inhibitive effectsionotropic GABAA receptororthosteric ‘GABA’ binding site

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