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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Synthesis of oxazolo-annulated 3-benzazepines designed by merging two negative allosteric NMDA receptor modulators

Alexander Markus1, Dirk Schepmann1, Bernhard Wünsch1,2

  • 1Institut für Pharmazeutische und Medizinische Chemie der Universität Münster, Münster, Germany.

Archiv Der Pharmazie
|February 28, 2022
PubMed

Keywords:
GluN2B subunitNMDA receptorbenzoxazolone bioisostereselimination of trifluoromethylsulfinateintramolecular Friedel-Crafts acylationtrifluoromethylsulfonyl protective group

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