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Updated: Sep 6, 2025

Monitoring GPCR-β-arrestin1/2 Interactions in Real Time Living Systems to Accelerate Drug Discovery
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Emerging structural insights into GPCR-β-arrestin interaction and functional outcomes.

Jagannath Maharana1, Ramanuj Banerjee1, Manish K Yadav1

  • 1Department of Biological Sciences and Bioengineering, Indian Institute of Technology, Kanpur 208016, India.

Current Opinion in Structural Biology
|June 23, 2022
PubMed
Summary

Recent studies reveal how β-arrestins (βarrs) interact with G protein-coupled receptors (GPCRs). Understanding these structural mechanisms is key to GPCR signaling and functional outcomes.

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