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Updated: Sep 6, 2025

Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay

Published on: February 28, 2025

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Discovery of the First-in-Class G9a/GLP Covalent Inhibitors

Kwang-Su Park1, Yan Xiong1, Hyerin Yim1

  • 1Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences, Oncological Sciences and Neuroscience, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.

Journal of Medicinal Chemistry
|June 28, 2022
PubMed

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