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Updated: Sep 1, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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Synthesis and biological testing of 3,5-bis(arylidene)-4-piperidone conjugates with

Margarita E Neganova1, Yulia R Aleksandrova1, Natalia S Nikolaeva2

  • 1Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, Moscow 119991, Russia; Institute of Physiologically Active Compounds, Russian Academy of Sciences, Chernogolovka 142432, Russia.

Bioorganic & Medicinal Chemistry Letters
|August 14, 2022
PubMed

Keywords:
1,2,3-Triazole1,2-OxaphospholeneAntitumor activityGlycolysisHeterocyclesPhosphorus“Click” chemistry

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