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Updated: Aug 31, 2025

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Single-Disulfide Conopeptide Czon1107, an Allosteric Antagonist of the Human α3β4 Nicotinic Acetylcholine Receptor

Yuan Ma1, Qiushi Cao1, Mengke Yang1

  • 1Key Laboratory of Marine Drugs, Chinese Ministry of Education, School of Medicine and Pharmacy, Ocean University of China, 5 Yushan Road, Qingdao 266003, China.

Marine Drugs
|August 25, 2022
PubMed

Keywords:
ACh-evoked currentsallosteric inhibitorconopeptidemolecular dynamics simulationsnAChRstructure–activity relationship

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