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The first structure-activity relationship study of oxytocin as a positive allosteric modulator for the µ opioid

Takaaki Mizuguchi1, Kanako Miyano2, Risa Yamauchi3

  • 1Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan; Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.

Peptides
|November 8, 2022
PubMed

Keywords:
AnalgesicsCyclic peptideOxytocinPositive allosteric modulatorμ Opioid receptor

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