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Updated: Aug 22, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Cardiovascular GPCR regulation by regulator of G protein signaling proteins

Anastasios Lymperopoulos1, Malka S Suster1, Jordana I Borges1

  • 1Laboratory for the Study of Neurohormonal Control of the Circulation, Department of Pharmaceutical Sciences, Nova Southeastern University College of Pharmacy, Fort Lauderdale, FL, United States.

Progress in Molecular Biology and Translational Science
|November 10, 2022
PubMed

Keywords:
ArrhythmiasCardiac myocyteCardiovascular diseaseG protein subunitG protein-coupled receptorHeart failurePlateletRegulator of G protein signalingSignal transductionVascular

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