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Updated: Aug 20, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Small-molecule allosteric inhibitors of GPX4

Hengrui Liu1, Farhad Forouhar2, Annie J Lin3

  • 1Department of Chemistry, Columbia University, New York, NY 10027, USA.

Cell Chemical Biology
|November 24, 2022
PubMed

Keywords:
GPX4allostericcancercysteinedrug discoveryenzymeglutathioneinhibitorperoxidasesmall molecule

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