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High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines
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Current Challenges in Small Molecule Proximity-Inducing Compound Development for Targeted Protein Degradation Using

Sridhar Radhakrishnan1, Oskar Hoff1, Markus K Muellner1

  • 1Celeris Therapeutics, Inc., Menlo Park, CA 94025, USA.

Molecules (Basel, Switzerland)
|December 11, 2022
PubMed

Keywords:
E3 ligaseE3 recruiterPICPROTACproximity-inducing compoundtargeted protein degradationubiquitination

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