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A Direct, Early Stage Guanidinylation Protocol for the Synthesis of Complex Aminoguanidine-containing Natural Products
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Guanidine Additive Enabled Intermolecular ortho-Phthalaldehyde-Amine-Thiol Three-Component Reactions for Modular

Carina Hey Pui Cheung1, Tin Hang Chong1, Tongyao Wei1

  • 1Department of Chemistry, State Key Laboratory of Synthetic Chemistry, The University of Hong Kong, Hong Kong SAR, P. R. China.

Angewandte Chemie (International Ed. in English)
|January 9, 2023
PubMed

Keywords:
ChemoselectivityDrug ConjugationIsoindolesOrtho-PhthalaldehydePeptide Conjugation

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