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Updated: Aug 12, 2025

Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay

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Structural insights into the potency and selectivity of covalent pan-FGFR inhibitors

Lingzhi Qu1, Xiaojuan Chen1, Hudie Wei2

  • 1Department of Oncology, NHC Key Laboratory of Cancer Proteomics, State Local Joint Engineering Laboratory for Anticancer Drugs, Xiangya Hospital, Central South University, Changsha, 410008, Hunan, China.

Communications Chemistry
|January 25, 2023
PubMed

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