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Updated: Aug 7, 2025

The Use of a β-lactamase-based Conductimetric Biosensor Assay to Detect Biomolecular Interactions
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The Use of a β-lactamase-based Conductimetric Biosensor Assay to Detect Biomolecular Interactions

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LY2183240 regioisomers act as competitive and selective inhibitors of class C β-lactamases

Pedro Ernesto de Resende1, Sarah Soares1, Mire Zloh1

  • 1UCL School of Pharmacy, Research Department of Pharmaceutical and Biological Chemistry, University College London, London, UK.

International Journal of Antimicrobial Agents
|March 9, 2023
PubMed

Keywords:
Antimicrobial resistanceCompetitive inhibitorLY2183240Tetrazoleβ-lactamases

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