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Updated: Jul 23, 2025

Electrophoretic Delivery of γ-aminobutyric Acid GABA into Epileptic Focus Prevents Seizures in Mice
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Electrophoretic Delivery of γ-aminobutyric Acid GABA into Epileptic Focus Prevents Seizures in Mice

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Three-Step Synthesis of the Antiepileptic Drug Candidate Pynegabine

Yi-Jing Sun1,2, Ya-Ling Gong1, Shi-Chao Lu1

  • 1State Key Laboratory of Bioactive Substance and Function of Natural Medicines and Beijing Key Laboratory of Active Substance Discovery and Druggability Evaluation, Institute of Materia Medica, Chinese Academy of Medical Sciences and Peking Union Medical College, 2A Nanwei Road, Xicheng District, Beijing 100050, China.

Molecules (Basel, Switzerland)
|July 14, 2023
PubMed

Keywords:
Buchwald–Hartwig cross couplingantiepileptic drugpynegabine

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