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N-Pyrazinylhydroxybenzamides as biologically active compounds: a hit-expansion study and antimicrobial evaluation

Marek Kerda1, Petr Šlechta1, Ondrej Jand'ourek1

  • 1Faculty of Pharmacy in Hradec Králové, Charles University, Hradec Králové, 500 05, Czech Republic.

Future Medicinal Chemistry
|October 25, 2023
PubMed

Keywords:
antibacterialantimicrobial resistanceantimycobacterialhit expansionmacromolecular assaymembrane depolarizationminimum bactericidal concentrationstructure–activity relationshipwater solubility

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