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Linkers as Game-changers in PROTAC Technology: Emphasizing General Trends in PROTAC Pharmacokinetics for their

Carlotta Cecchini1,2, Sébastien Tardy3,2, Leonardo Scapozza4,2

  • 1Pharmaceutical Biochemistry/Chemistry, School of Pharmaceutical Sciences, University of Geneva, Rue Michel-Servet 1, CH-1206 Geneva. carlotta.cecchini@unige.ch.

Chimia
|December 9, 2023
PubMed

Keywords:
Drug metabolism and pharmacokineticsLinker optimizationProteolysis Targeting Chimeras (PROTACs)Targeted protein degradation

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