Related Experiment Video

Updated: Jun 19, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Molecular mechanism of the endothelin receptor type B interactions with Gs, Gi, and Gq

Donghee Ham1, Wataru Shihoya2, Osamu Nureki2

  • 1School of Pharmacy, Sungkyunkwan University, 2066 Seobu-ro, Jangan-gu, Suwon 16419, Republic of Korea.

Structure (London, England : 1993)
|July 23, 2024
PubMed

Keywords:
ET(B)G proteinHDX-MSconformationsignal selectivity

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