A review on tyrosine kinase inhibitors for targeted breast cancer therapy

Vidya Sankarapandian1, Ramya Lakshmi Rajendran2, Conrad Ondieki Miruka3

  • 1Department of Microbiology and Immunology, Kampala International University, Western Campus, Box 20000, Uganda.

PubMed

Insights

Tyrosine kinase inhibitors (TKIs) are effective targeted therapies for breast cancer, disrupting tumor growth pathways. This review explores TKIs in clinical trials, showing improved survival and potential for personalized breast cancer treatment.

Area of Science:

  • Oncology
  • Molecular Biology
  • Pharmacology

Background:

  • Breast cancer is a complex disease with molecular heterogeneity.
  • Overexpressed tyrosine kinase receptors are linked to poor prognosis, making them therapeutic targets.
  • Tyrosine kinase inhibitors (TKIs) disrupt key pathways in tumor growth and proliferation.

Purpose of the Study:

  • To review current and emerging tyrosine kinase inhibitors (TKIs) for breast cancer treatment.
  • To explore the role of TKIs in preclinical studies and clinical trials.
  • To discuss the integration of TKIs into personalized breast cancer therapy.

Main Methods:

  • Literature review of preclinical studies and clinical trials on TKIs in breast cancer.
  • Analysis of TKI mechanisms targeting receptor tyrosine kinases (e.g., HER2, EGFR, VEGFR).
  • Examination of TKI efficacy when used in combination with chemotherapy, endocrine therapy, or other targeted agents.

Main Results:

  • TKIs targeting various tyrosine kinases (HER2, EGFR, VEGFR, ALK, RET, FGFR, ROS1, MAPK, TRK) are crucial in breast cancer.
  • Approved TKIs like lapatinib, neratinib, and tucatinib improve progression-free and overall survival.
  • TKIs show promise as a therapeutic option for various breast cancer subtypes.

Conclusions:

  • TKIs represent a significant advancement in targeted breast cancer therapy.
  • Combination therapies involving TKIs enhance patient outcomes.
  • Future breast cancer treatment will likely involve novel TKIs and personalized strategies.

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