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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay

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Exploring covalent inhibitors of SARS-CoV-2 main protease: from peptidomimetics to novel scaffolds

Noor Atatreh1,2, Radwa E Mahgoub1,2, Mohammad A Ghattas1,2

  • 1College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emirates.

Journal of Enzyme Inhibition and Medicinal Chemistry
|February 6, 2025
PubMed

Keywords:
Anti-viralCovid-19covalent inhibitorirreversible inhibitionwarheads reactivity

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