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Updated: May 13, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Thienopyrimidinone Derivatives as a GluN2B/C/D Biased, Positive Allosteric Modulator of the N-Methyl-d-Aspartate

Russell G Fritzemeier1, Nicholas S Akins1, Paul J Arcoria1

  • 1Department of Chemistry, Emory University, Atlanta, Georgia 30322, United States.

Journal of Medicinal Chemistry
|April 21, 2025
PubMed

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