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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Catalyzed Asymmetric Michael Additions of 1-Pyrroline Esters with β-Fluoroalkyl Alkenyl Imides and Azodicarboxylates

De-Hua Zhang1, Yi-Chao Li1, Jin-Chen You1

  • 1Hubei Key Laboratory of Nanomedicine for Neurodegenerative Diseases, School of Chemistry, Chemical Engineering and Life Science, Wuhan University of Technology, Wuhan, 430070, China.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|May 7, 2025
PubMed

Keywords:
1‐Pyrroline estersasymmetric michael additionsazodicarboxylatesβ‐fluoroalkyl alkenyl imides

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