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Continuous Flow Chemistry: Reaction of Diphenyldiazomethane with p-Nitrobenzoic Acid
Published on: November 15, 2017
John M Saunders1, Esveidy Oceguera Nava1, Jason Li1
1Department of Chemistry & Biochemistry, University of California, Santa Barbara, California 93106, United States.
A novel recyclable coupling agent, 2,2'-dipyridyldithiocarbonate (DPDTC), enables efficient synthesis of thioesters and amides in a plug flow reactor (PFR). This method offers high yields for diverse acid and amine couplings, including peptides.
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