Targeting anti-apoptosis as a therapeutic strategy in neuroendocrine neoplasms

PubMed

Insights

Venetoclax, a BCL-2 inhibitor, showed a partial response in a pancreatic neuroendocrine tumor (pNET) patient. High BCL2 expression in neuroendocrine neoplasms (NENs) correlates with aggressive features and poorer survival.

Area of Science:

  • Oncology
  • Molecular Biology
  • Genetics

Background:

  • Anti-apoptotic protein BCL-2 is expressed in aggressive neuroendocrine neoplasms (NENs).
  • Venetoclax targets BCL-2 and is used for chronic lymphocytic leukemia treatment.

Purpose of the Study:

  • To report a case of pancreatic neuroendocrine tumor (pNET) treated with venetoclax.
  • To characterize BCL2 expression in a large cohort of NENs and correlate it with clinical and molecular features.

Main Methods:

  • Case report of a pNET patient treated with venetoclax.
  • Next-generation sequencing (DNA and RNA) of 636 NENs (pancreatic, small bowel, colorectal, lung).
  • Comparison of BCL2 expression in NENs versus non-NEN cancers and correlation with MKI67, mutations, survival, and immune markers.

Main Results:

  • The pNET patient achieved a partial response to venetoclax lasting 30 months.
  • Colorectal, lung, and pancreatic NENs showed higher BCL2 expression than non-NENs.
  • BCL2-high NENs were associated with higher MKI67, increased RB1 mutations in pNETs, decreased overall survival, and enriched immune microenvironment.

Conclusions:

  • This is the first reported case of a pancreatic NET responding to venetoclax.
  • BCL2 expression is a marker of aggressive NENs, associated with poor prognosis and an immune-enriched tumor microenvironment.

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