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Updated: Sep 15, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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A Structure-Activity Relationship Study of Novel Positive Allosteric Modulators for the δ-Opioid Receptor

Owindeep Deo1, Vi Pham2, Sadia Alvi2

  • 1Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.

ACS Chemical Neuroscience
|July 18, 2025
PubMed
Abstract

Keywords:
allosteric modulatorbiased modulationchronic painoperational model of allosterismstructure−activity relationshipδ-opioid receptor

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