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Unraveling the therapeutic landscape of approved non-peptide macrocycles

Zhonghua Li1, Zhenqiang Zhang1, Bin Yu2,3

  • 1Academy of Chinese Medical Sciences, Collaborative Innovation Center of Research and Development on the Whole Industry Chain of Yu-Yao, Henan University of Chinese Medicine, Zhengzhou 450046, China.

Acta Pharmaceutica Sinica. B
|July 23, 2025
PubMed

Keywords:
Drug discoveryMacrocyclesMacrocyclizationMolecular editingNon-peptides

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