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Structural Basis of PPARγ-Mediated Transcriptional Repression by the Covalent Inverse Agonist FX-909

Zane T Laughlin1, Liudmyla Arifova1,2, Paola Munoz-Tello1

  • 1Department of Biochemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Journal of Medicinal Chemistry
|August 13, 2025
PubMed
Abstract

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