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Updated: Sep 11, 2025

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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Beyond purinergic signaling: Dual ligand approaches to multitarget drug discovery

Beatrice Francucci1, Aleksei Smirnov1, Andrea Spinaci1

  • 1School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, Via Madonna delle Carceri, 62032 Camerino, Italy.

Drug Discovery Today
|August 17, 2025
PubMed

Keywords:
A(2A) adenosine receptorsdual ligandsmultitargets compoundspurinergic receptors

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