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Updated: Jan 13, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

11.8K

Research towards selective inhibition of the CLK3 kinase

Vinay Kumar Singh1,2, Frédéric Justaud1, Dabbugoddu Brahmaiah3

  • 1Univ Rennes, CNRS, ISCR (Institut des Sciences Chimiques de Rennes), UMR 6226, F-35000 Rennes, France.

Beilstein Journal of Organic Chemistry
|October 29, 2025
PubMed

Keywords:
CLK3cancerkinasesmolecular modellingquinazolinestriazoles

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