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Updated: Jan 11, 2026

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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A New Era for PPARγ: Covalent Ligands and Therapeutic Applications

Jasmine L King1, Luke Smithers1, Alice Vrielink1

  • 1School of Molecular Sciences, The University of Western Australia, Crawley, 6009 Perth, Australia.

Journal of Medicinal Chemistry
|November 11, 2025
PubMed
Abstract

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