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The Development of UM-203, A Reversible Covalent STING Antagonist

Leonard Barasa1,2, Leo DeOrsey1,2, Maeve D O'Reilly1,2

  • 1Program in Chemical Biology, University of Massachusetts Chan Medical School, 364 Plantation Street, Worcester, Massachusetts 01605, United States.

ACS Medicinal Chemistry Letters
|January 14, 2026
PubMed
Abstract

Keywords:
CytokinesOligomerizationStimulator of interferon genesTBK1Type I interferoninhibitor

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