Related Experiment Video

Updated: Jan 16, 2026

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay
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Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay

Published on: December 19, 2018

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Structural Pharmacology of Estrogen-Related Receptors

Puhan Zhao1,2, Hong Fang1,3, Bahaa Elgendy1,3,2

  • 1Center for Clinical Pharmacology, Washington University School of Medicine in St. Louis and University of Health Sciences & Pharmacy in St. Louis, St. Louis, Missouri 63110, United States.

ACS Pharmacology & Translational Science
|January 15, 2026
PubMed

Keywords:
conformational dynamicsestrogen related receptors (ERRs)inverse agonists and selective modulatorsligand-binding domain (LBD) structurenuclear receptor pharmacologystructural basis of receptor function

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