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Updated: Jun 22, 2026

Solid Phase Synthesis of a Functionalized Bis-Peptide Using "Safety Catch" Methodology
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Solid Phase Synthesis of a Functionalized Bis-Peptide Using "Safety Catch" Methodology

Published on: May 15, 2012

Efficient Synthesis of Enlicitide Chloride through Convergent Solution-Phase and Hybrid Solution-Solid-Phase

Xuting Zhao1, Xinqi Li1, Shuxian Zhang1

  • 1Department of Medicinal Chemistry, Shandong Key Laboratory of Druggability Optimization and Evaluation for Lead Compounds, School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong 250012, China.

Precision Chemistry
|March 27, 2026
PubMed
Abstract

Keywords:
PCSK9 inhibitorchemical synthesisenlicitidehybrid solution−solid-phase strategymacrocyclic peptide

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