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Updated: Apr 1, 2026

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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From Flat to 3D: Replacing Phenyl Rings with Saturated Bridged Bicyclic Mimetics to Mitigate Bioactivation and

Murugaiah A M Subbaiah1, Shruti Surendran2, Gaurav Saini3

  • 1Department of Medicinal Chemistry, Discovery and Development Sciences, Biocon Bristol Myers Squibb R&D Centre, Syngene, Bommasandra Phase IV, Jigani Link Road, Bengaluru 560099, India.

Journal of Medicinal Chemistry
|March 30, 2026
PubMed

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