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Quantitative Methods to Study Protein Arginine Methyltransferase 1-9 Activity in Cells
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Unique Cysteine-Directed Covalent Inhibition of PRMT1 Suppresses Breast Tumorigenesis

Min Shao1, Ruining Li1, Jinglei Hu1

  • 1Shanghai Frontiers Science Center of Targeted Drugs, State Key Laboratory of Innovative Immunotherapy, Shanghai Key Laboratory for Molecular Engineering of Chiral Drugs, Engineering Research Center of Cell & Therapeutic Antibody Ministry of Education, School of Pharmaceutical Sciences, Shanghai Jiao Tong University, Shanghai 200240, China.

Journal of Medicinal Chemistry
|June 17, 2026
PubMed
Abstract

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