Related Experiment Video

Updated: Aug 10, 2026

Structure-Guided Design and Development of Novel Cyclophilin A Inhibitors and Ganoderiol-F Derivatives: An In-Silico Approach
10:01

Structure-Guided Design and Development of Novel Cyclophilin A Inhibitors and Ganoderiol-F Derivatives: An In-Silico Approach

Published on: June 23, 2026

Design, synthesis, and biological activity of novel oxazole-based small molecule allosteric GLP-1R agonists

Ruifeng Wang1, Qing Liu2, Chaoyu Lu2

  • 1School of Pharmacy, Shanxi Medical University, Taiyuan, 030001, China; Department of Endocrinology, First Hospital of Shanxi Medical University, Shanxi Medical University, Taiyuan, Shanxi, 030001, China.

European Journal of Medicinal Chemistry
|August 8, 2026
PubMed

Keywords:
GLP-1 receptorOxazolePositive allosteric modulatorType 2 diabeteshGLP-1R KI mice

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