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Allosteric Crosstalk between Inhibitor Binding Sites Drives Enhanced Islatravir Susceptibility in F227C HIV-1 Reverse

Corey W Hecksel1, Susanne N Walker1, Izzat Raheem2

  • 1Department of Protein & Structural Chemistry, Merck & Co., Inc., West Point, Pennsylvania19486, United States.

ACS Infectious Diseases
|September 11, 2026
PubMed

Keywords:
HIV-1 RTNNRTINRTTIcryoEMdoravirineislatravir

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