Related Experiment Video

Updated: Oct 3, 2026

High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines
05:33

High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines

Published on: November 9, 2020

Vepdegestrant: the first FDA-approved oral PROTAC and a milestone in targeted protein degradation

Jeffrey Yang1, Longqin Hu2,3

  • 1Hansoh Bio, LLC, 9900 Medical Center Drive, Suite 200, Rockville, MD, 20850, USA. jeffrey.yang@hansohbio.com.

Medicinal Chemistry Research : an International Journal for Rapid Communications on Design and Mechanisms of Action of Biologically Active Agents
|October 1, 2026
PubMed

Keywords:
Breast cancerERαEstrogen receptorPROTACTargeted protein degradationVepdegestrant

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