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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
07:30

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

Synthesis of Substituted Indazoles With Potential Kinase Inhibitory Activity

Achraf Hibot1, Abderrafia Hafid2, Mostafa Khouili2

  • 1Laboratory of Medicinal Chemistry, Department of Pharmacology, Toxicology and Medicinal Chemistry, Faculty of Pharmacy and Food Sciences, University of Barcelona, Barcelona, Spain.

Chemmedchem
|October 9, 2026
PubMed

Keywords:
C‐arylationN‐arylationSuzuki–Miyauracross‐couplingindazole

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