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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Sulfonyl-Imidazopyridines Decouple Reactivity from Stability for Ligandability Mapping and Covalent Inhibitor

Zhihong Li1, Madeleine L Ware1, Phillip W Gingrich2

  • 1Department of Chemistry, University of Texas at Austin, Austin, Texas78712, United States.

Journal of the American Chemical Society
|October 27, 2026
PubMed

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