Structural themes of cereblon-recruiting degraders: selected recent examples

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High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines
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High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines

Published on: November 9, 2020

Sana Ahmed1, Michael Rowley1

  • 1Department of Biochemistry and Molecular Biology, University of British Columbia, Vancouver, BC V6T 1Z3, Canada.

Acta Crystallographica. Section F, Structural Biology Communications
|November 6, 2026
PubMed

Keywords:
PROTACsX-ray crystallographycerebloncryo-EMmolecular-glue degradersstructural biologystructure-based drug design

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