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Potency and maintenance requirement of atracurium and vecuronium given alone or together

P Rautoma1, O Erkola, O A Meretoja

  • 1Maria Hospital, University of Helsinki, Finland.

Insights

Combining atracurium and vecuronium muscle relaxants in adults demonstrates significant potentiation, reducing overall drug consumption by approximately 30%. This combination offers an intermediate-acting effect for neuromuscular blockade maintenance during anesthesia.

Area of Science:

  • Anesthesiology
  • Pharmacology
  • Neuromuscular Blockade

Background:

  • Synergistic effects are known for some competitive muscle relaxants.
  • Previous studies on muscle relaxant combinations primarily focused on pediatric patients.

Purpose of the Study:

  • To evaluate the maintenance requirement and synergistic effects of combining atracurium and vecuronium in adult surgical patients.
  • To determine the dose-response relationship and potential drug savings with a combined agent.

Main Methods:

  • 45 adult surgical patients (ASA I-II) received propofol-alfentanyl-N2O-O2 anesthesia.
  • Individual dose-response curves were established for atracurium and vecuronium in 30 patients.
  • 15 patients received a combination of atracurium and vecuronium (cAV) in equipotent ratios.

Main Results:

  • ED95 values were 260 ± 9 µg/kg for atracurium and 59 ± 3 µg/kg for vecuronium.
  • The combination (cAV) showed significant potentiation (P = 0.0001), with an ED95 of 94 ± 7 µg/kg atracurium and 21 ± 2 µg/kg vecuronium.
  • Maintenance requirements for cAV were 120 µg/kg/h atracurium and 27 µg/kg/h vecuronium, a 30% reduction in drug consumption.

Conclusions:

  • Atracurium and vecuronium exhibit significant synergism in adult patients, maintaining potentiation throughout anesthesia.
  • The combination acts as an intermediate-acting muscle relaxant.
  • Using the atracurium-vecuronium combination can reduce overall drug consumption by approximately 30%.

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