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Bioorganic & Medicinal Chemistry Letters|March 17, 2018
Discovery of a highly potent orally bioavailable imidazo-[1, 2-a]pyrazine Aurora inhibitorTao Yu, Yonglian Zhang, Angela D Kerekes, et al.Bioorganic & Medicinal Chemistry Letters|January 7, 2012
The discovery of potent, selective, and orally active pyrazoloquinolines as PDE10A inhibitors for the treatment of SchizophreniaGinny D Ho, Shu-Wei Yang, Jennifer Smotryski, et al.Bioorganic & Medicinal Chemistry Letters|June 13, 2020
Discovery of hydroxy pyrimidine Factor IXa inhibitorsCharles L Jayne, Teresa Andreani, Tin-Yau Chan, et al.Bioorganic & Medicinal Chemistry Letters|April 15, 2017
Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitorsIsao Sakurada, Toshiya Endo, Katsuyoshi Hikita, et al.Journal of Medicinal Chemistry|June 23, 2016
Discovery of 1-(1H-Pyrazolo[4,3-c]pyridin-6-yl)urea Inhibitors of Extracellular Signal-Regulated Kinase (ERK) for the Treatment of CancersJongwon Lim, Elizabeth H Kelley, Joey L Methot, et al.ACS Medicinal Chemistry Letters|March 18, 2026
<i>N</i>‑Alkyl and <i>N</i>‑Aryl Aminopyrazole Spirocarbamates: A Two-Pronged Lead Optimization Strategy to Identify Orally Bioavailable Plasma Kallikrein InhibitorsRohan R Merchant, Natalia Chernyak, Jovan A Lopez, et al.ACS Chemical Biology|February 8, 2018
Discovery of Selective RNA-Binding Small Molecules by Affinity-Selection Mass SpectrometryNoreen F Rizvi, John A Howe, Ali Nahvi, et al.Bioorganic & Medicinal Chemistry Letters|May 5, 2015
Rapid development of two factor IXa inhibitors from hit to leadDann L Parker, Shawn Walsh, Bing Li, et al.Bioorganic & Medicinal Chemistry Letters|May 17, 2015
Development of a novel class of potent and selective FIXa inhibitorsTing Zhang, Patrick Andre, Thomas J Bateman, et al.ACS Medicinal Chemistry Letters|June 6, 2014
Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine CoreTao Yu, Jayaram R Tagat, Angela D Kerekes, et al.Pageof 3